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LINDA STREET, PHD
PHD
Clinical Psychologist
NPI: 1184225849Individual
Specialties, Licenses & Credentials
Research & Publications (20)
Optimisation of a series of potent, selective and orally bioavailable GlyT1 inhibitors.
PMID 19318248·Bioorg Med Chem Lett·2009
4-observational
2,3,7-Trisubstituted pyrazolo[1,5-d][1,2,4]triazines: functionally selective GABAA alpha3-subtype agonists.
PMID 16621541·Bioorg Med Chem Lett·2006
8-other
Discovery of imidazo[1,2-b][1,2,4]triazines as GABA(A) alpha2/3 subtype selective agonists for the treatment of anxiety.
PMID 16480260·J Med Chem·2006
7-preclinical
Imidazo[1,2-a]pyrimidines as functionally selective GABA(A) ligands.
PMID 16406613·Bioorg Med Chem Lett·2006
8-other
Imidazo[1,2-a]pyrimidines as functionally selective and orally bioavailable GABA(A)alpha2/alpha3 binding site agonists for the treatment of anxiety disorders.
PMID 16392789·J Med Chem·2006
7-preclinical
Imidazo[1,2-b][1,2,4]triazines as alpha2/alpha3 subtype selective GABA A agonists for the treatment of anxiety.
PMID 16386900·Bioorg Med Chem Lett·2006
7-preclinical
Imidazo[1,2-a]pyrazin-8-ones, imidazo[1,2-d][1,2,4]triazin-8-ones and imidazo[2,1-f][1,2,4]triazin-8-ones as alpha2/alpha3 subtype selective GABA A agonists for the treatment of anxiety.
PMID 16384707·Bioorg Med Chem Lett·2006
7-preclinical
Spectroscopic phase-dispersion optical coherence tomography measurements of scattering phantoms.
PMID 19529186·Opt Express·2006
8-other
TPA023 [7-(1,1-dimethylethyl)-6-(2-ethyl-2H-1,2,4-triazol-3-ylmethoxy)-3-(2-fluorophenyl)-1,2,4-triazolo[4,3-b]pyridazine], an agonist selective for alpha2- and alpha3-containing GABAA receptors, is a nonsedating anxiolytic in rodents and primates.
PMID 16183706·J Pharmacol Exp Ther·2006
7-preclinical
7-(1,1-Dimethylethyl)-6-(2-ethyl-2H-1,2,4-triazol-3-ylmethoxy)-3-(2-fluorophenyl)-1,2,4-triazolo[4,3-b]pyridazine: a functionally selective gamma-aminobutyric acid(A) (GABA(A)) alpha2/alpha3-subtype selective agonist that exhibits potent anxiolytic activity but is not sedating in animal models.
PMID 16279764·J Med Chem·2005
7-preclinical
Data courtesy of the U.S. National Library of Medicine (NLM). Ltrl is not affiliated with or endorsed by NLM.
Contact & Hours
- Address
- 165 SAINT REGIS DR
MASSAPEQUA PARK, NY 11762 - Phone
- (516) 672-6746
Quick Facts
- NPI
- 1184225849
- Entity Type
- Individual
- Gender
- Female
- Medicare
- Not confirmed
- Specialties
- 1
- Locations
- 1
- Publications
- 20
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